A Phase I, Open-Label, Multi-Center, First-in-Human Trial to Investigate E303, in Participants With Advanced Refractory Solid Tumors
Summary
This is a Phase I trial to evaluate the safety, tolerability and efficacy of nectin-4 targeting antibody-drug conjugate (SBE303) in participants with advanced solid tumors
Arms & interventions
- DrugE303
All participants will receive an intravenous (IV) infusion of E303
Outcome measures
Primary
Incidence of adverse events and serious adverse events
Time frame: Until trial completion (estimated 3 years)
Incidence of dose limiting toxicity
Time frame: For the first cycle of treatment, through pre-dose Cycle 2 Day 1
Confirmed objective response rate
Efficacy enpoint per Blinded Independent Central Review (BICR), according to Response Evaluation Criteria in Solid Tumors (RECIST) v1.1
Time frame: 32 weeks
Secondary
Tumor response
Time frame: 32 weeks
Disease control rate
Time frame: 32 weeks
Area under the plasma/serum concentration vs time curve of total E303
Time frame: Until trial completion (estimated 3 years)
Maximum plasma/serum concentration of total E303
Time frame: Until trial completion (estimated 3 years)
Time to reach maximum plasma/serum concentration of total E303
Time frame: Until trial completion (estimated 3 years)
Plasma/serum concentration before the next dose of total E303
Time frame: Until trial completion (estimated 3 years)
Terminal half life of total E303
Time frame: Until trial completion (estimated 3 years)
Incidence and titer of anti-drug antibodies
Time frame: Until trial completion (estimated 3 years)
Incidence of neutralizing antibodies
Time frame: Until trial completion (estimated 3 years)
Eligibility criteria
Study locations (2)
Research Site
Scottsdale, Arizona, 85258
Research Site
Fairfax, Virginia, 22031