A Phase 1, First-in-human, Dose Escalation Study of JNJ-95804306 for Relapsed or Refractory Hematological Malignancies
Summary
The purpose of Part 1 (Dose Escalation) of the study is to assess how safe and tolerable JNJ-95804306 is and to find out the most suitable dose (recommended phase 2 dose \[RP2D\]) of JNJ-95804306. The purpose of Part 2 (Dose Expansion) is to further assess the safety of JNJ-95804306 and determine the anti-tumor activity alone and/or when administered in addition to standard of care (SoC) therapy at the putative RP2D(s) regimens in participants with hematological malignancies (cancer that begins in blood-forming tissue, such as the bone marrow, or in the cells of the immune system). For US sites: The purpose of Part 1 (Dose Escalation) of the study is to assess how safe and tolerable JNJ-95804306 is and to find out the most suitable dose (recommended phase 2 dose \[RP2D\]) of JNJ-95804306. The purpose of Part 2 (Dose Expansion) is to further assess the safety of JNJ-95804306 and determine the anti-tumor activity alone at the putative RP2D(s) regimens in participants with hematological malignancies (cancer that begins in blood-forming tissue, such as the bone marrow, or in the cells of the immune system).
Arms & interventions
- DrugJNJ-95804306
JNJ-95804306 will be administered orally.
- DrugAML SoC
AML SoC will be administered subcutaneously/intravenously.
- DrugCLL/SLL SoC
CLL/SLL SoC will be administered orally/ intravenously.
Outcome measures
Primary
Part 1: Number of Participants with Dose Limiting Toxicities (DLTs)
A DLT is defined as any toxicity that requires discontinuation of treatment; any Grade 5 toxicity; Non-hematologic Toxicity (Grade 3 or 4); and unacceptable hematologic toxicity.
Time frame: Up to 21 days after first full dose of study drug
Number of Participants with Adverse Events (AEs) by Severity
An AE is any untoward medical occurrence in a participant administered a pharmaceutical (investigational or non investigational) product. An AE does not necessarily have a causal relationship with the treatment. Severity of AEs will be graded according to the National Cancer Institute Common Terminology Criteria for Adverse Events (NCI-CTCAE) version (v) 6.0. by using standard grades as follows: Grade 1: Mild; asymptomatic or mild symptoms; Grade 2: Moderate; minimal, local or noninvasive intervention indicated; Grade 3: Severe but not immediately life threatening; hospitalization or prolongation of hospitalization indicated; Grade 4: Life-threatening consequences; and Grade 5: Death related to AE.
Time frame: Up to 6 years 5 months
Secondary
For US sites: Part 1: Number of Participants with Dose Limiting Toxicities (DLTs)
Time frame: Up to first 28 days after first dose of study drug
Serum Concentrations of JNJ-95804306
Time frame: Up to approximately 6 years 5 months
Area Under the Curve From Time of Administration until End of Dosing Interval (AUC[t]) of JNJ-95804306
Time frame: Up to approximately 6 years 5 months
Maximum Plasma Concentration (Cmax) of JNJ-95804306
Time frame: Up to approximately 6 years 5 months
Minimum Plasma Concentration (Cmin) of JNJ-95804306
Time frame: Up to approximately 6 years 5 months
Complete Response (CR) in Participants with Acute Myeloid Leukemia (AML)
Time frame: Up to 6 years 5 months
Overall Response (OR) in Participants with Myelodysplastic Syndrome (MDS)
Time frame: Up to 6 years 5 months
Complete Response (CR) in Participants with MDS
Time frame: Up to 6 years 5 months
Overall Response (OR) in Participants with Chronic Lymphocytic Leukemia (CLL)
Time frame: Up to 6 years 5 months
Complete Response in Participants with CLL
Time frame: Up to 6 years 5 months
Overall Response in Participants with Small Lymphocytic Lymphoma (SLL)
Time frame: Up to 6 years 5 months
Complete Response in Participants with SLL
Time frame: Up to 6 years 5 months
Duration of Response (DoR)
Time frame: Up to 6 years 5 months
Time to Response (TTR)
Time frame: Up to 6 years 5 months
Eligibility criteria
Study locations (3)
Indiana Blood & Marrow Transplantation
Indianapolis, Indiana, 46237
Start Midwest
Grand Rapids, Michigan, 49546
Rutgers Cancer Institute of New Jersey
Piscataway, New Jersey, 08854